In stock
Retatrutide peptid 10mg
119,00€
Trojni agonist hormonskih receptorjev, ki cilja na receptorje GIP, GLP-1 in glukagon, proučevan v sodobnih presnovnih raziskavah.
Opis
Retatrutide peptid 10mg za raziskovalno uporabo
Retatrutide je raziskovalni peptid naslednje generacije s trojnim delovanjem (agonist receptorjev GLP-1, GIP in glukagona), ki se proučuje zaradi njegove vloge pri uravnavanju presnove, signalizaciji apetita in raziskavah telesne sestave.
Raziskane lastnosti
- Trojni agonist receptorjev (GLP-1 / GIP / glukagon)
- Raziskan za napredne presnovne poti in poti izgube maščobe
- Proučevan za uravnavanje apetita in porabe energije
Čistost in dokumentacija
Vsaka viala Retatrutide 10mg je HPLC-preverjena z več kot 99-odstotno čistostjo, pridobljena v skladu z GMP in opremljena s celotno dokumentacijo za laboratorijske raziskave.
Raziščite več spojin v naši kategoriji Peptidi za hujšanje in izgubo maščobe. Vsi izdelki se prodajajo izključno za laboratorijske in raziskovalne namene ter niso namenjeni za uporabo pri ljudeh.
Pregled raziskav
Retatrutide je sintetični peptid z 39 aminokislinami, ki predstavlja vrhunec raziskav metabolizma na več receptorjih. Kot uravnotežen trojni agonist receptorjev GIP, GLP-1 in glukagona hkrati vključuje tri ločene hormonske poti.
Komponenta GLP-1 spodbuja od glukoze odvisno izločanje inzulina in centralni občutek sitosti; komponenta GIP krepi odzive trebušne slinavke in modulira delovanje adipocitov; dodana komponenta glukagona pa aktivira porabo energije v jetrih in oksidacijo lipidov — mehanizem, ki ga monoagonisti GLP-1 in dvojni agonisti GIP/GLP-1, kot je Tirzepatide, nimajo.
Retatrutide, zasnovan z lipidnim delom z dikislino maščobne kisline C20 za vezavo na albumin, doseže raziskavam prijazno razpolovno dobo približno 6 dni. Raziskovalci ga uporabljajo za proučevanje energijskega ravnovesja, jetrne steatoze, telesne sestave, lipidomskih profilov in medsebojnega delovanja receptorjev za inkretin/glukagon. Z zgodnjimi predkliničnimi in kliničnimi podatki, ki kažejo na najboljše učinke v svojem razredu na telesno težo in metabolne markerje, Retatrutide hitro postaja referenčna molekula za raziskave metabolizma s trojnimi agonisti.
Raziskovalne uporabe
- Študije interakcij na treh receptorjih
- Raziskave porabe energije
- Napredna analiza metabolnih poti
- Študije oksidacije lipidov
Tehnične specifikacije
| CAS številka | 2381089-83-2 |
|---|---|
| Molekulska formula | C221H343N51O63 |
| Molarna masa | 4731.45 g/mol |
| Sekvenca / Struktura | Trojni agonist GIP/GLP-1/Glucagon (39 aminokislin, modificiran s C20 maščobno dikislino) |
| Sinonimi | LY3437943 |
| Razpolovna doba | Približno 6 dni |
| Topnost | Topno v bakteriostatični vodi |
| Čistost | 99%+ testirano s HPLC |
| Oblika | Liofiliziran prašek, 10mg / vialo |
| Koda izdelka | RT10 |
Ravnanje in shranjevanje
Shranjujte liofilizirano pri -20°C. Po rekonstituciji hranite v hladilniku pri 2 do 8°C in porabite v roku 21 dni.
- Rekonstituirajte izključno s sterilnim topilom raziskovalne kakovosti v skladu z vašim laboratorijskim protokolom.
- Izogibajte se ponavljajočim se ciklom zamrzovanja in odmrzovanja ter zabeležite datum rekonstitucije, koncentracijo in temperaturo shranjevanja.
- Namenjeno izključno za in-vitro raziskave ali kvalificirane laboratorijske delovne procese.

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